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ibicuruzwa

Uruganda rukora ifu ya Galantamine Hydrobromide No. CAS: 1953-04-4 Ubuziranenge bwa 98% ku bikoresho by'inyongera

Ibisobanuro bigufi:

Ni ubwoko bwa benzozepine bukomoka ku tubuto n'indabyo bya narcissus, osmanthus, cyangwa canna. Ni kandi umuti ubuza kolinesterase mu kanwa.


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Ibirango by'ibicuruzwa

Ibipimo by'ibicuruzwa

Izina ry'igicuruzwa Galantamine Hydrobromide
Irindi zina Galanthamine hydrobromide;

Galantamine HBr;

Galanthamine HBr; (4aS, 6R, 8aS) -4a, 5,9,10,11,12-hexahydro-3-mikorerexy-11-methyl-6H-Benzofuro

Nimero ya CAS 1953-04-4
Ifishi y'ingirabuzimafatizo C17H21NO3.HBr
Uburemere bwa molekile 368.27
Ubwiza 98.0%
Isura ifu y'umweru kuva kuri umweru kugeza kuri umweru
Gupakira 1kg/umufuka 10kgs, 25kgs/ingoma
Porogaramu imiti ya nootropic

Intangiriro y'ibicuruzwa

Galantamine hydrobromide ni benzazepine ikomoka ku tubuto n'indabyo bya narcissus, osmanthus, cyangwa canna. Ni kandi umuti ubuza kolinesterase mu kanwa. Nk'umusemburo w'uduce twa acetylcholine twa nicotinic, yakoreshejwe cyane mu kunoza imikorere y'ubwonko. Inshingano yayo ni ukubuza kolinesterase mu buryo buhanitse kandi bugasubira inyuma, bityo yongera urugero rwa acetylcholine. Iyo galantamine hydrobromide yinjijwe mu maraso, yinjizwa mu bice bitandukanye by'umubiri, harimo n'ubwonko. Ifatana na receptor za nicotinic acetylcholine, igatera impinduka mu miterere yayo no kongera irekurwa rya acetylcholine. Ikora kandi mu guhangana no gusubiza inyuma ingaruka z'uduce twa kolinesterase. Mu kubuza kolinesterase, irinda gusenyuka kwa acetylcholine, bityo yongera urugero n'igihe cy'iyi neurotransmitter ikomeye. Galantamine ishobora kandi kunoza imyigire no kwibuka, ikarinda ububyimbirwe bw'ubwonko, kandi ikabungabunga urugero rwo hejuru rw'uduce twa neurotransmitters binyuze mu kubungabunga ubusugire bwa neuron na synapses.

Ikiranga

Galantamine Hydrobromide

(1) Ubuziranenge bwinshi: Galantamine hydrobromide ishobora kuba umusaruro utunganye cyane binyuze mu gutunganya ikorwa ryayo. Ubuziranenge bwinshi busobanura ko binyabuzima biboneka neza kandi ingaruka mbi zikaba nke.

(2) Umutekano: Byagaragaye ko Galantamine hydrobromide ari umuti utekanye ku mubiri w'umuntu.

(3) Gutuza: Galantamine hydrobromide ifite gutuza neza kandi ishobora gukomeza imikorere yayo n'ingaruka zayo mu bidukikije bitandukanye no mu buryo butandukanye bwo kubika.

Porogaramu

Nk'inyongeramusaruro, galantamine hydrobromide ishobora kunoza kwibuka, ubwenge, n'ubushobozi bwo gukora imirimo ya buri munsi. Ikora mu kugarura uburinganire bw'ibintu bimwe na bimwe karemano (neurotransmitters) mu bwonko, byongera umuvuduko wo kwibuka no kunoza kubika amakuru n'ibintu bifatika. Byongeye kandi, galantamine hydrobromide igira ingaruka ku buryo butaziguye cyangwa butaziguye ku mikorere y'ubwonko. Itera imbaraga mu buryo butaziguye mu mikorere ya synaptic binyuze mu gukora microglia na astrocytes. Galantamine itanga uburinzi ku mikorere ya antioxydant iterwa na radicals free.

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