Galantamine Hydrobromide ikora ifu ya CAS No.: 1953-04-4 98% isuku min.kubintu byongeweho
Ibipimo byibicuruzwa
Izina RY'IGICURUZWA | Galantamine Hydrobromide |
Irindi zina | Hydrobromide ya Galanthamine; Galantamine HBr; Galanthamine HBr; (4aS, 6R, 8aS) -4a, 5,9,10,11,12-hexahydro-3-imikorere-11-methyl-6H-Benzofuro [3a, 3,2-ef] 6-ol, Hydrobromide |
URUBANZA No. | 1953-04-4 |
Inzira ya molekulari | C17H21NO3.HBr |
Uburemere bwa molekile | 368.27 |
Isuku | 98.0% |
Kugaragara | cyera kugeza ifu yera |
Gupakira | 1kg / umufuka 10kgs, 25kgs / ingoma |
Gusaba | nootropics |
Kumenyekanisha ibicuruzwa
Hydrobromide ya Galantamine ni ubwoko bwa benzozepine ikomoka ku matara n'indabyo za narcissus, osmanthus, cyangwa canna.Ninumunwa wa cholinesterase munwa.Nka ligande ya nicotinic acetylcholine reseptor, yakoreshejwe cyane mugutezimbere imikorere ya neurocognitive.Uruhare rwarwo ni uguhiganwa no guhindagura acetylcholinesterase, bityo bikongerera ingufu za acetylcholine.
Iyo yinjiye mumaraso, hydrobromide ya galanthamine yinjira byoroshye mubice byose byumubiri, harimo nubwonko.Ihuza na reseptor ya nicotinic acetylcholine, itera impinduka zifatika kandi ikarekura acetyloline.Irakora kandi mukurushanwa no guhindura ingaruka za cholinesterase inhibitor.Muguhagarika cholinesterase, irinda kwangirika kwa acetyloline, bityo bikongerera urwego nigihe kirekire cyiyi neurotransmitter ikomeye.Galanthamine kandi itezimbere ubushobozi bwo kwiga no kwibuka, ikumira ubwonko kandi ikagumana urugero rwinshi rwa neurotransmitter ikomeza ubusugire bwa neuron na synaps
Ikiranga
.Yongera umuvuduko wo kwibuka no kunoza kugumana amakuru arambuye.
(2) Ubushobozi bwo kwiga butezimbere mukwongera plastike ya synaptic na neuroplastique.Hydrobromide ya Galanthamine itaziguye cyangwa itaziguye igira ingaruka kuri neuroplastique.Itera synaptic ya plastike ikora microglia na astrocyte.
(3) Ifasha gusinzira kandi byongera kuruhuka.Galanthamine irashobora kongera ingorane zo gusinzira itera gusinzira vuba amaso, bityo bigatuma ibitotsi byiyongera.
.Irashobora kurinda selile yubwonko kwangirika kwa okiside kugirango igumane imikorere myiza yubwonko.