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ibicuruzwa

Galantamine Hydrobromide ikora ifu ya CAS No.: 1953-04-4 98% isuku min.kubintu byongeweho

Ibisobanuro bigufi:

Nubwoko bwa benzozepine ikomoka kumatara nindabyo za narcissus, osmanthus, cyangwa canna.Ninumunwa wa cholinesterase munwa.


Ibicuruzwa birambuye

Ibicuruzwa

Ibipimo byibicuruzwa

Izina RY'IGICURUZWA Galantamine Hydrobromide
Irindi zina Hydrobromide ya Galanthamine;

Galantamine HBr;

Galanthamine HBr; (4aS, 6R, 8aS) -4a, 5,9,10,11,12-hexahydro-3-imikorere-11-methyl-6H-Benzofuro [3a, 3,2-ef] 6-ol, Hydrobromide

URUBANZA No. 1953-04-4
Inzira ya molekulari C17H21NO3.HBr
Uburemere bwa molekile 368.27
Isuku 98.0%
Kugaragara cyera kugeza ifu yera
Gupakira 1kg / umufuka 10kgs, 25kgs / ingoma
Gusaba nootropics

Kumenyekanisha ibicuruzwa

Hydrobromide ya Galantamine ni ubwoko bwa benzozepine ikomoka ku matara n'indabyo za narcissus, osmanthus, cyangwa canna.Ninumunwa wa cholinesterase munwa.Nka ligande ya nicotinic acetylcholine reseptor, yakoreshejwe cyane mugutezimbere imikorere ya neurocognitive.Uruhare rwarwo ni uguhiganwa no guhindagura acetylcholinesterase, bityo bikongerera ingufu za acetylcholine.

Iyo yinjiye mumaraso, hydrobromide ya galanthamine yinjira byoroshye mubice byose byumubiri, harimo nubwonko.Ihuza na reseptor ya nicotinic acetylcholine, itera impinduka zifatika kandi ikarekura acetyloline.Irakora kandi mukurushanwa no guhindura ingaruka za cholinesterase inhibitor.Muguhagarika cholinesterase, irinda kwangirika kwa acetyloline, bityo bikongerera urwego nigihe kirekire cyiyi neurotransmitter ikomeye.Galanthamine kandi itezimbere ubushobozi bwo kwiga no kwibuka, ikumira ubwonko kandi ikagumana urugero rwinshi rwa neurotransmitter ikomeza ubusugire bwa neuron na synaps

Ikiranga

.Yongera umuvuduko wo kwibuka no kunoza kugumana amakuru arambuye.

(2) Ubushobozi bwo kwiga butezimbere mukwongera plastike ya synaptic na neuroplastique.Hydrobromide ya Galanthamine itaziguye cyangwa itaziguye igira ingaruka kuri neuroplastique.Itera synaptic ya plastike ikora microglia na astrocyte.

(3) Ifasha gusinzira kandi byongera kuruhuka.Galanthamine irashobora kongera ingorane zo gusinzira itera gusinzira vuba amaso, bityo bigatuma ibitotsi byiyongera.

.Irashobora kurinda selile yubwonko kwangirika kwa okiside kugirango igumane imikorere myiza yubwonko.

Porogaramu

Hydrobromide ya Galantamine irashobora kunoza kwibuka, ubwenge, nubushobozi bwo gukora imirimo ya buri munsi.Ikora mukugarura uburinganire bwibintu bimwe na bimwe (neurotransmitters) mubwonko.


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