Ifu ya Nefiracetam ikora CAS No.: 77191-36-7 99% isuku min. kubintu byongeweho
Video y'ibicuruzwa
Ibipimo byibicuruzwa
| Izina ryibicuruzwa | Nefiracetam |
| Irindi zina | n- (2,6-dimethylphenyl) -2-oxo-1-pyrrolidineacetamide; NEFIRACETAM; 2-oxo-1-pyrrolidinylaceticacid, 2,6-dimethylanilide; dm9384; n- (2,6-dimethylphenyl) -2-oxo-1-pyrrolidineacetamid; DM-9384, (2- (2-Oxopyrrolidin-1-yl) -N- (2,6-dimethylphenyl) -acetamide); DMMPA |
| URUBANZA No. | 77191-36-7 |
| Inzira ya molekulari | C14H18N2O2 |
| Uburemere bwa molekile | 246.3 |
| Isuku | 99.0% |
| Kugaragara | Ifu yera |
| Gupakira | 25 kg / barrale |
| Gusaba | nootropic |
Kumenyekanisha ibicuruzwa
Nefiracetam ni iyumuryango wa piracetam, icyiciro cyibiyobyabwenge bizwiho kwongera ubwenge. Nefiracetam yashizwemo bwa mbere mu ntangiriro ya za 1980 kandi yahise ikurura abantu kubera uburyo bwihariye bwibikorwa hamwe nibishobora kuvurwa. Ivanguramoko rishingiye ku moko ritekereza ko rigira ingaruka kuri neurotransmitter na reseptors mu bwonko, amaherezo rikazamura ubushobozi bwubwenge. Nefiracetam yibasira cyane ubwonko bwa acetylcholine, urufunguzo rwingenzi rwa neurotransmitter ishinzwe kwibuka, kwiga, hamwe nibikorwa byubwenge. Muguhindura reseptor ya acetylcholine, nefiracetam ituma itumanaho ryiyongera hagati ya neuron, bityo bikazamura plastike ya synaptic no kunoza imitekerereze. Byongeye kandi, nefiracetam ikorana na acide ya gamma-aminobutyric (GABA) kugirango ifashe kuringaniza imiterere ya neurotransmitter. Mu kugira ingaruka nziza no kubuza neurotransmitters, nefiracetam ifasha kugumana imikorere myiza yubwonko, bityo igateza imbere kwibanda, kwitabwaho, hamwe nibikorwa rusange byubwenge.
Ikiranga
(1) Isuku ryinshi: Nefiracetam irashobora kubona ibicuruzwa byera cyane binyuze mugutunganya umusaruro. Isuku ryinshi risobanura bioavailable nziza hamwe na reaction nkeya.
(2) Umutekano: Umutekano mwinshi, reaction nkeya.
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Porogaramu
Nefiracetam ni hydrophobique ikomoka kuri piracetam, ubusanzwe ifatwa nkibintu bishinzwe kuvumbura imiyoboro ya calcium mu mubiri no guhererekanya mu buryo butaziguye ibintu byerekana ibimenyetso bishimishije nka agoniste igice cyimiyoboro ya calcium ion. Glycine ihuza urubuga rwa reseptor ya NDMA. Binyuze mu ngaruka zayo ku bwonko bwubwonko, nefiracetam irashobora kongera ubushobozi bwubwenge kandi ikarinda kwiga no kutagira ubwenge. Ntabwo ifite imitekerereze ya muscarinic agonist cyangwa antagonist, ntanubwo ibuza ibikorwa bya acetylcholinease. Kubwibyo rero, ingaruka zayo zo kurwanya amnestic no kongera imbaraga zo kwibuka zigerwaho mugutezimbere irekurwa rya acetyloline mu bwonko bwubwonko.
