Amino Tadalafil ikora ifu CAS No.: 385769-84-6 98% isuku min.kubintu byongeweho
Ibipimo byibicuruzwa
| Izina RY'IGICURUZWA | Amino Tadalafil |
| Irindi zina | . (6R, 12aR) -2-Amino-6- 3,4-b] indole-1,4-dione; AminoTadalafil (6R, 12Ar) -2-Amino-6- (1,3-Benzodioxol-5-Yl) -2,3,6,7,12,12A -Hexahydropyrazino [1 ', 2': 1,6] Pyrido [3,4-B] Indole-1,4-Dione; (6R, 12aR) -2-Amino-6- (benzo [d] [1,3 dioxol-5-yl) -2,3,6,7,12,12a-hexahydropyrazino [1 ', 2': 1,6] pyrido [3,4-b] indol-1,4-dione; (6R , 12aR) -2-amino-6- (benzo [d] [1,3] dioxol-5-yl) -2,3,12,12a-tetrahydropyrazino [1 ', 2': 1,6] pyrido [3 , 4-b] indole-1,4 (6H, 7H) -dione |
| URUBANZA No. | 385769-84-6 |
| Inzira ya molekulari | C21H18N4O4 |
| Uburemere bwa molekile | 390.39 |
| Isuku | 98.0% |
| Kugaragara | Ifu yera-yera |
| Gusaba | Ibyokurya byongera ibiryo |
Kumenyekanisha ibicuruzwa
Amino Tadalafil ni uruganda rusa na Tadalafil, hamwe na hamwe mumatsinda akora mumiterere yarwo asimburwa nitsinda rya amino.Nibikoresho bya PDE5 kandi bifite ingaruka za farumasi zisa na Tadalafil.Ikoreshwa cyane cyane mukuvura imikorere mibi yumugabo (ED).Ugereranije na Tadalafil, Amino Tadalafil ifite umuvuduko muke wa metabolike mu mubiri, bityo bikaba bishobora kugira ingaruka ndende.
Ikiranga
.Ibi bivuze ko Amino Tadalafil ishobora guhagarika neza imikorere ya enzyme ya PDE5, igatera umuvuduko wamaraso mubice byimyororokere yumugabo no kunoza ibimenyetso byimikorere mibi (ED).
.Ibi bituma Amino Tadalafil akora imiti myinshi yo kuvura ED, idakenera gufatwa kenshi.
(3) Ingaruka nkeya: Amino Tadalafil ifite ingaruka nke ugereranije na Tadalafil, nko kubabara umutwe, no kubura gastrointestinal.Bitewe no guhitamo kwinshi, Amino Tadalafil irashobora kwirinda neza imikoranire nubundi bwoko bwa PDE, bikagabanya ingaruka zingaruka.
.Ibi bituma Amino Tadalafil afite ibyifuzo byinshi byo gusaba mugihe kizaza.
Porogaramu
Amino Tadalafil ni uruganda rwateye imbere mumyaka yashize, rufite imiterere isa na Tadalafil, ariko amatsinda amwe mumiterere yayo asimburwa nitsinda rya amino.Kugeza ubu, Amino Tadalafil ntabwo yemerewe gukoreshwa mu buvuzi, bityo ikoreshwa ryayo mu buvuzi ni rito.Nyamara, ubushakashatsi bumwe bwerekanye ko iyi nteruro ifite amahirwe menshi yo gushyira mubikorwa.
Amino Tadalafil ni inhibitor ya PDE5, ifite ingaruka za farumasi nka Tadalafil.Irashobora kunoza ibimenyetso byimikorere idahwitse (ED) iteza imbere umuvuduko wamaraso mubice byimyororokere yumugabo muguhagarika ibikorwa bya enzyme ya PDE5.Ugereranije na Tadalafil, Amino Tadalafil ifite umuvuduko wa metabolisme gahoro mu mubiri, ishobora kugira ingaruka zirambye.Ibi bituma Amino Tadalafil afite amahirwe menshi yo kuvura ED.
Byongeye kandi, Amino Tadalafil irashobora kandi gukoreshwa mu kuvura izindi ndwara zimwe na zimwe, nka hypertension yimpyiko.Ubushakashatsi bumwe bwerekanye ko inhibitori ya PDE5 ishobora kwagura imiyoboro yamaraso, bityo bikazamura ibimenyetso byabarwayi bafite hypertension yimpyiko.Kubera ko Amino Tadalafil ifite imiti isa na Tadalafil, irashobora no gukoreshwa mu kuvura hypertension yimpyiko.
Muri rusange, Amino Tadalafil ifite amahirwe menshi yo gukoreshwa, ariko harakenewe ibigeragezo byinshi byamavuriro kugirango umenye umutekano wacyo.Niba ibi bigeragezo bitanga umusaruro ushimishije, Amino Tadalafil irashobora kuba imiti mishya yo kuvura hypertension ya ED na pulmonary arterial hypertension, itanga uburyo bwinshi bwo kuvura abaganga n’abarwayi n’abaganga.
