page_banner

ibicuruzwa

Uruganda rukora ifu ya Coluracetam CAS No.: 135463-81-9 99% isuku min.kubintu byongeweho

Ibisobanuro bigufi:

Coluracetam ni umwe mu bagize umuryango wa racetam w’ibintu bya nootropique kandi uzwi kandi nka MKC-231.Yakozwe na Kobe Pharmaceutical Company mu Buyapani hagamijwe kuvura AD nubumuga bwo kutamenya.


Ibicuruzwa birambuye

Ibicuruzwa

Ibipimo byibicuruzwa

Izina RY'IGICURUZWA

Coluracetam

Irindi zina

MKC-231;

2-oxo-N- (5,6,7,8-tetrahydro-2,3-dimethyl-furo [2,3-b] quinolin-4-yl) -1-pyrrolidineacetamide

URUBANZA No.

135463-81-9

Inzira ya molekulari

C19H23N3O3

Uburemere bwa molekile

341.4

Isuku

99.0%

Kugaragara

Ifu yera

Gusaba

Ibyokurya byongera ibiryo

Kumenyekanisha ibicuruzwa

Coluracetam ni umwe mu bagize umuryango wa racetam w’ibintu bya nootropique kandi uzwi kandi nka MKC-231.Yakozwe na Kobe Pharmaceutical Company mu Buyapani hagamijwe kuvura AD nubumuga bwo kutamenya.

Uburyo nyabwo bwibikorwa bya Coluracetam ntabwo bwumvikana neza, ariko byizera ko bukora cyane muguhindura sisitemu ya cholinergique.Byatekerejweho kongera urugero rwa acetylcholine, urufunguzo rwingenzi rwa neurotransmitter mubwonko bufitanye isano rya bugufi no kwiga no kwibuka.Coluracetam irashobora kubigeraho yongera umubare nigikorwa cyabatwara choline itwara abantu, biganisha ku kurekura kwa acetyloline no kurushaho gukwirakwiza ibimenyetso hagati ya neuron.

Nubwo ubushakashatsi kuri Coluracetam bugifite aho bugarukira, ubushakashatsi bwakozwe hakiri kare hamwe nubushakashatsi bwinyamanswa bwerekanye ingaruka zishobora gutera neuroprotective na cognitive-kongera imbaraga.Ubushakashatsi bumwe bwerekanye ko Coluracetam ifite iterambere runaka mubumuga bwo kwibuka muburyo bwa AD.

Kubijyanye nubushakashatsi bwamavuriro, ubushakashatsi kuri Coluracetam bwibanze ahanini kubushakashatsi bwinyamaswa ndetse nigeragezwa ryabantu.Harakenewe ubushakashatsi nibimenyetso byinshi kugirango umenye umutekano wacyo nibikorwa byabantu.Kugeza ubu, Coluracetam ntabwo yemerewe gukoreshwa mu mavuriro, ariko ikoreshwa cyane nk'inyongera ya nootropique yo kongera ubumenyi mu bihugu bimwe na bimwe.

Kubireba umutekano, hari amakuru make yubushakashatsi aboneka ku ngaruka n'ingaruka z'igihe kirekire za Coluracetam.Ukurikije ubumenyi buriho, Coluracetam muri rusange ifatwa nkaho ifite umutekano, ariko birasabwa kugisha inama inzobere mu by'ubuzima, cyane cyane niba ufite ubuzima bwiza cyangwa ufata indi miti, mbere yo kuyikoresha.

Muncamake, Coluracetam nikintu cya nootropic kirimo kwigwa kubushobozi bwacyo mukuvura AD nubumuga bwo kutamenya.Mugihe ubushakashatsi bwambere bwerekana ko ubwenge bwiyongera ningaruka za neuroprotective, harakenewe ubushakashatsi bwinshi kugirango hamenyekane neza umutekano wacyo.

Ikiranga

.Uku kwera kwinshi bigira uruhare mu kunoza bioavailable kandi bigabanya kubaho kwimyitwarire mibi.

(2) Umutekano: Coluracetam ifatwa nkumutekano kubyo kurya byabantu.Ubushakashatsi bwagutse bwerekanye ubumara bwabwo buke hamwe ningaruka ntoya murwego rusabwa.

.Uku gushikama kwemeza imikorere ihamye kandi yizewe mugihe runaka.

(4) Absorption Byihuse: Coluracetam yakirwa byoroshye numubiri wumuntu.Iyo umaze kwinjizwa, byinjira vuba mumaraso unyuze mumara kandi bigakwirakwizwa neza mubice bitandukanye ningingo zitandukanye, bikorohereza ingaruka zifuzwa.

(5) Kuzamura ubumenyi: Coluracetam izwiho ubushobozi bwo kuzamura imikorere yubwenge, harimo kunoza kwibuka, ubushobozi bwo kwiga, no kwibanda.Bikunze gushakishwa nabantu bashaka kunoza imikorere yabo yo mumutwe.

.

.Nyamara, ubushakashatsi buracyakenewe kugirango twumve neza akamaro kayo mukuvura ibi bihe byihariye.

Porogaramu

Kuri ubu Coluracetam irakoreshwa mubikorwa bitandukanye kandi yerekana ibyiringiro by'ejo hazaza.Ikoreshwa cyane cyane nk'inyongera yo kongera ubwenge, ishakishwa nabantu bashaka kunoza imitekerereze yabo, kwibanda, hamwe nubushobozi bwo kwiga.Ubushobozi bwikomatanya bwo guhindura sisitemu ya cholinergique bizera ko bigira uruhare mubikorwa byayo byongera ubwenge.

Usibye ubu ikoreshwa muri iki gihe, Coluracetam yerekanye ubushobozi mu kuvura indwara zifata ubwonko nk'indwara ya Alzheimer n'ubumuga bwo kutamenya.Ubushakashatsi bwerekana ko Coluracetam ishobora kuba ifite imitekerereze ya neuroprotective, bigatuma iba umukandida ushishikajwe no gukora ubushakashatsi muri ibi bihe.Nyamara, ubushakashatsi bwimbitse hamwe nubuvuzi burakenewe kugirango hamenyekane imikorere yacyo, umutekano, hamwe na protocole ikoreshwa neza mumavuriro.

Abaturage bageze mu za bukuru bongereye icyifuzo cyo gutabara gishobora kugabanya kugabanuka kwubwenge.Ingaruka za neuroprotective ya Coluracetam hamwe nubushobozi bwo gushyigikira uburyo bwo gusana imitsi bituma iba inzira ishimishije yubushakashatsi mugukemura ikibazo cyo kugabanuka kwubwenge bujyanye no gusaza.

Byongeye kandi, ubushakashatsi bwibanze bwerekana ko Coluracetam ishobora kugira inyungu kubibazo byo guhungabana nko kwiheba no guhangayika.Nyamara, ubushakashatsi bwimbitse burasabwa gusuzuma imikorere yacyo no gushyiraho protocole ikwiye yo kuvura muri ibi bimenyetso.

Ubushobozi bwa Coluracetam bugera no muri gahunda ya neurorehabilitation nayo.Ubushobozi bwayo bwo kongera ibimenyetso bya neuronal kandi birashobora gushyigikira uburyo bwo gusana imitsi bituma iba umukandida kugirango akoreshwe mu gusubiza mu buzima busanzwe abantu bafite ibikomere cyangwa ubwonko.

Mugihe Coluracetam yerekana amasezerano mubikorwa bitandukanye, ni ngombwa gushimangira ko hakenewe ubundi bushakashatsi, kwemeza imikorere yayo, umutekano, hamwe na protocole ikoreshwa neza.Ibyemezo byemewe nabyo bizakenerwa kugirango bikoreshe ivuriro mubimenyetso byihariye.


  • Mbere:
  • Ibikurikira:

  • Andika ubutumwa bwawe hano hanyuma utwohereze