Ifu ya Sunifiram Nomero ya CAS: 314728-85-3 Isuku ya 99% ku bikoresho by'inyongera
Videwo y'ibicuruzwa
Ibipimo by'ibicuruzwa
| Izina ry'igicuruzwa | Sunifiram |
| Irindi zina | 1-(4-Benzoylpiperazin-1-yl)propan-1-imwe; 1-Benzoyl-4-(1-oxopropyl)piperazine |
| Nimero ya CAS | 314728-85-3 |
| Ifishi y'ingirabuzimafatizo | C14H18N2O2 |
| Uburemere bwa molekile | 246.30 |
| Ubwiza | 99.0% |
| Isura | ifu y'umweru ya kristu |
| Gupakira | 1kg/umufuka |
| Porogaramu | imiti ya nootropic |
Intangiriro y'ibicuruzwa
Sunifiram ni umuti wa AMPA receptor agonist wongera ubushobozi bwo gutanga amakuru kuri receptor za AMPA mu bwonko, akenshi bifatwa nk'ibifite uruhare runini mu kwiga no kwibuka. Mu kongera imikorere ya receptor za AMPA, Sunifiram ifatwa nk'ifasha mu kongera ubushobozi bwo kwiga no kwibuka mu bwonko, ndetse inanoza ubushobozi bwo gutekereza no gushyira mu gaciro. Byongeye kandi, ikora mu gukangura imikorere ya receptor za glutamate no kongera umusaruro no kurekura acetylcholine ya "learning neurotransmitter". Sunifiram ikora cyane cyane nk'ikintu cya ampa, bivuze ko ihuzwa na receptor za glutamate zo mu bwoko bwa AMPA mu bwonko nyuma yo kwambuka umupaka w'amaraso n'ubwonko. Ibi bitera imbaraga mu gukora glutamate, neurons y'ingenzi mu gutuma synaptic plasticity, cyangwa ubushobozi bwa synapses z'imitsi bwo gusubiza kwiyongera cyangwa kugabanuka kw'ibikorwa. Urugero rwa Glutamate ni ingenzi cyane muri hippocampus, igice cy'ubwonko gikora uruhare runini mu kugenda mu kirere, kwibuka no kubika. Urugero rwa glutamate ruhagije ni ingenzi mu kongera cyangwa kunoza ibimenyetso mu gihe kirekire hagati y'imitsi. Imbaraga ni ingenzi. Ingufu nyinshi za Sunifilaram zongerera ubushobozi bwo gutekereza zikora binyuze mu kongera imbaraga z'ibimenyetso by'ubwonko muri iki gice cy'ubwonko.
Ikiranga
(1) Ubuziranenge bwinshi: Sunifiram ishobora kubona ibicuruzwa bifite ubuziranenge bwinshi binyuze mu buryo bwo gukora bunoze. Ubuziranenge bwinshi busobanura ko binyabuzima biboneka neza kandi ingaruka mbi zikaba nke.
(2) Umutekano: Byagaragaye ko Sunifiram ari umuti utekanye ku mubiri w'umuntu.
(3) Gutuza: Sunifiram ifite ubutuza bwiza kandi ishobora gukomeza imikorere yayo n'ingaruka zayo mu bidukikije bitandukanye no mu buryo butandukanye bwo kubika.
Porogaramu
Sunifiram ni umuti wongera ubushobozi bwo gutekereza, uboneka kandi nk'inyongera mu mirire, utekerezwaho kunoza imikorere y'ubwonko no kunoza imyigire n'ubwitonzi. Ukora binyuze mu gutunganya za receptor za AMPA mu bwonko. AMPA ni urwego rw'imitsi rufasha mu gutumanaho vuba hagati y'uturemangingo two mu bwonko. Ituma umuntu yihuta cyane mu myigire, kwibuka no kwibuka, ndetse no kunoza uburyo yitonze, gushishikarira no gusobanukirwa neza ibintu.












