Ifu ya Nefiracetam ikora CAS No.: 77191-36-7 99% isuku min.kubintu byongeweho
Ibipimo byibicuruzwa
| Izina RY'IGICURUZWA | Nefiracetam |
| Irindi zina | n- (2,6-dimethylphenyl) -2-oxo-1-pyrrolidineacetamide; NEFIRACETAM; 2-oxo-1-pyrrolidinylaceticacid, 2,6-dimethylanilide; dm9384; n- (2,6-dimethylphenyl) -2-oxo-1-pyrrolidineacetamid; DM-9384, (2- (2-Oxopyrrolidin-1-yl) -N- (2,6-dimethylphenyl) -acetamide); DMMPA |
| URUBANZA No. | 77191-36-7 |
| Inzira ya molekulari | C14H18N2O2 |
| Uburemere bwa molekile | 246.3 |
| Isuku | 99.0% |
| Kugaragara | Ifu yera |
| Gupakira | 25 kg / barrale |
| Gusaba | nootropic |
Kumenyekanisha ibicuruzwa
Nefiracetam ni iy'ubwenge butagira umupaka bwongera urwego rw'ibiyobyabwenge, bifite imiterere itandukanye ya chimique kandi byongera ubushobozi bwubwenge kandi bikarinda kwangirika kwimyigire no kwibuka binyuze mu ngaruka zabyo ku bwonko bwubwonko.Ntabwo ifite imiterere ya muscarinic reseptor agonist na antagonist, ntanubwo ibuza ibikorwa bya Ach.Ingaruka zo kurwanya kwibagirwa no kongera imbaraga muri uyu muti zigerwaho no kongera irekurwa rya Ach mu bwonko bwubwonko.Intungamubiri zishingiye kuri protein kinase zongera ibikorwa bya Ca2 + umuyoboro, zishobora kuba inshingano zo kuzamura Ach kurekura.Nefiracetam (NEF) ni ubwoko bwa pyrrolidone nootropic agent hamwe na farumasi zitandukanye kimwe ningaruka zongera ubumenyi.Mu gufatwa na amygdala, nefiracetam irabuza gufata electroencephalographic ndetse no gufata imyitwarire.NEF ifite antikonvulsant itandukanye.
Ikiranga
Nefiracetam ikoreshwa mu kuvura indwara zifata ubwonko.Irashobora kongera ubushobozi bwubwenge kandi ikarinda kwangirika kwimyigire no kwibuka bitewe n'ingaruka zayo kuri cortex.Ntabwo ifite imiterere ya muscarinic reseptor agonist na antagonistic agent, ntanubwo ibuza ibikorwa bya acetyl cholinase.Kubwibyo, kurwanya kwayo kwibagirwa no kongera imbaraga yibuka bibaho mugutezimbere irekurwa rya acetylcholine mumyanya yubwonko.
Porogaramu
Nefiracetam ni hydrophobique ikomoka kuri piracetam hamwe na synthèse synthique ya Racetam yose ivanze piracetam.Nefiracetam ikorwa cyane cyane na Daiichi Sankyo (uruganda rukora imiti mu Buyapani) kugirango ivure AD.Usibye uburyo bwose bwitiriwe Nefiracetam generally muri rusange bikekwa ko ari ibintu bishinzwe kuvumbura imiyoboro ya calcium mu mubiri, ndetse no guhererekanya mu buryo butaziguye ibintu byerekana ibimenyetso bishimishije, bikora nka agoniste igice cya glycine-ihuza urubuga rwa reseptor ya NDMA.
