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ibicuruzwa

Ingano ya CAS y'umusaruro w'ifu wa PRL-8-53: 51352-87-5 98% by'ubuziranenge bw'ibicuruzwa by'inyongera

Ibisobanuro bigufi:

PRL-8-53 ni umuti mushya wongera ubushobozi bwo gutekereza, ukaba ari ikintu kirinda uturemangingo tw’imitsi. Wakozwe bwa mbere na Dr. Milton V.


Ibisobanuro birambuye ku gicuruzwa

Ibirango by'ibicuruzwa

Ibipimo by'ibicuruzwa

Izina ry'igicuruzwa

PRL-8-53

Irindi zina

Methyl 3-(2-(benzyl(Methyl)aMino)ethyl)benzoate hydrochloride;aside Benzoic, 3-[2-[methyl(phenylmethyl)amino]ethyl]-, ester ya methyl, hydrochloride (1:1);Methyl 3-{2-[benzyl(methyl)amino]ethyl}benzoate hydrochloride (1:1)

Nimero ya CAS

51352-87-5

Ifishi y'ingirabuzimafatizo

C18H22ClNO2

Uburemere bwa molekile

319.83

Ubwiza

98.0%

Isura

Ifu y'umweru

Gupakira

1 kg kuri buri gafuka 25kg / ingoma

Porogaramu

nootropic

Intangiriro y'ibicuruzwa

PRL-8-53, izwi kandi nka methyl 3-(2-(benzyl(methyl)amino)ethyl)benzoate, ni ikintu cyakozwe mu buryo bwa nootropic gitekerezwaho kugira ngo cyongere ikwirakwizwa rya kolinergic kandi kigenzura urugero rwa dopamine mu bwonko. Izi myitwarire zigira uruhare mu ngaruka zayo zishobora kongera ubushobozi bwo gutekereza, bityo bikanoza imiterere y'ubuhanga, kubika no kugarura ibintu. Ubushakashatsi bwinshi ku nyamaswa n'abantu bwagaragaje ibisubizo byiza ku miterere yayo yo kongera kwibuka. Mu bushakashatsi bwakozwe ku buryo bworoshye kandi bugenzurwa na placebo, abantu bahawe dose imwe ya PRL-8-53 bagaragaje ubushobozi bwo kwibuka no kugarura amagambo neza ugereranije n'itsinda rya placebo. Ibi byavumbuwe byateye amatsiko n'ubushakashatsi bwinshi ku bushobozi bw'icyo kintu. Ubundi bushakashatsi bwakozwe ku mbeba bwagaragaje ko guha PRL-8-53 byazamuye cyane ubushobozi bwabyo bwo kwiga mu kazi ko mu mazi. Imbeba zavuwe na PRL-8-53 zashoboye kubona urubuga rwihishe neza kurusha uburyo bwo kuzigenzura, bigaragaza ubushobozi bw'icyo kintu nk'uburyo bwo kongera kwibuka.

Ikiranga

(1) Ubuziranenge buhanitse: PRL-8-53 ishobora kubona ibicuruzwa bifite ubuziranenge buhanitse binyuze mu gutunganya umusaruro. Ubuziranenge buhanitse busobanura ko binyabuzima biboneka neza kandi ingaruka mbi zikaba nke.

(2) Umutekano: Umutekano mwinshi, ingaruka mbi nke, nta ngaruka mbi zigaragara.

(3) Gutuza: PRL-8-53 ifite umutekano mwiza kandi ishobora gukomeza imikorere yayo n'ingaruka zayo mu bidukikije bitandukanye no mu buryo butandukanye bwo kubika.

Porogaramu

Nk'ubwoko bushya bw'inyongeramusaruro yo kongera ubushobozi bwo gutekereza, PRL-8-53 irushaho kunoza kwibuka by'igihe gito no kwibuka mu gihe gito, mu gihe yongera ubushobozi bwo kwiga no kwihuta mu kumenya ubumenyi, bigafasha mu kunoza imyigire no gukora neza. Ubushakashatsi bwerekana ko PRL-8-53 ishobora guteza imbere imikurire n'ivugururwa ry'imitsi yo mu bwonko. PRL-8-53 ishobora kongera umuvuduko ubwonko bukoresha mu gutunganya amakuru, bigatuma abantu barangiza imirimo no gufata ibyemezo vuba. Nubwo ugereranije n'izindi nyunganiramirire za nootropic Ariko, ubushakashatsi kuri PRL-8-53 ni buke, ariko ubushakashatsi buriho bugaragaza ko bufite ubushobozi bwo kunoza ubushobozi bwo kwibuka no gutekereza.


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