J-147 uruganda rukora ifu CAS No.: 1146963-51-0 99.0% isuku min.kubintu byongeweho
Ibipimo byibicuruzwa
Izina RY'IGICURUZWA | 2,2,2-Trifluoroacetic aside 1- (2,4-DiMethylphenyl) -2 - [(3-Methoxyphenyl) Methylene] hydrazide] |
Irindi zina | J-147, J147 |
URUBANZA No. | 1146963-51-0 |
Inzira ya molekulari | C18H17F3N2O2 |
Uburemere bwa molekile | 350.33 |
Isuku | 99% |
Kugaragara | Ifu yera |
Gupakira | 1kg kumufuka |
Gusaba | nootropics |
Kumenyekanisha ibicuruzwa
J-147 ni imbaraga zikomeye mu kanwa zikora neuroprotectant zikomoka cyane cyane kuri curcumin, ingirakamaro muri turmeric.Bitandukanye na curcumin, irenga inzitizi yamaraso-ubwonko neza.Muri byo, J-147 ikora ihuza na ATP synthase.Umusaruro mwinshi wa ATP ujyanye no gusaza.Usibye kongera urwego rwa neurotransmitters NGF na BDNF, J-147 irashobora kugenzura ibi.Byongeye kandi, J-147 ibuza monoamine oxydease B na transport ya dopamine.Guteza imbere ubwonko bwongera urwego rwo gukura kwimitsi (NGF) hamwe nubwonko bukomoka mubwonko (BDNF).Icy'ingenzi cyane, J-147 irashobora guteza imbere imikurire yimitsi mishya, kongera ubushobozi bwubwonko bwo kwiga no kwibuka, no kunoza imikorere yubwenge.
Ikiranga
(1) Isuku ryinshi: J-147 irashobora kubona ibicuruzwa bifite isuku nyinshi binyuze mu gutunganya umusaruro.Isuku ryinshi risobanura bioavailable nziza hamwe na reaction nkeya.
(2) Umutekano: J-147 byagaragaye ko ifite umutekano ku mubiri w'umuntu.
(3) Guhagarara: J-147 ifite ituze ryiza kandi irashobora gukomeza ibikorwa byayo n'ingaruka zayo ahantu hatandukanye no kubika.
(4) Biroroshye kubyakira: J-147 irashobora kwinjizwa vuba numubiri wumuntu, ikinjira mumaraso binyuze mumara, kandi igakwirakwizwa mubice bitandukanye.
Porogaramu
J-147 ni uruganda rukomatanya uburyo bwibanze bwibikorwa birimo kuzamura mitochondial, bityo bigatuma ingufu zitangwa ku rwego rwa selire.J-147 yashizweho kugirango yongere ubushobozi bwubwonko bwo gusana no kwirinda ibyangizwa nimyaka bitewe no kunoza imikorere ya mito-iyambere.Byongeye kandi, J-147 yerekana ibintu byingenzi birwanya anti-inflammatory na antioxydeant, bikarushaho kongera ingaruka ziterwa na neuroprotective.J-147 irashobora guteza imbere imikurire yingirabuzimafatizo nshya, kongera ubushobozi bwubwonko bwo kwiga no kwibuka, no kunoza imikorere yubwenge.